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Preclamol and parkinsonian fluctuationsPirtošek, Zvezdan, 1956- ...Preclamol, the (-)enantiomer of 3-PPP (=3(3-hydroxyphenyl)-N- n-propyl piperidine), has a selective dopamine autoreceptor- and postsynaptic mixed agonist-antagonist profile. Its action on patients ... with disabling on-off parkinsonian fluctuations has been studied and compared with those of placebo and subcutaneous apomorphine. Preclamol had a mild but unequivocal antiakinetic effect, less than that caused by subcutaneous apomorphine, but itprovoked less dyskinesia. Further studies to explore the therapeutic potential of preclamol seem justified.Vir: Clinical neuropharmacology. - ISSN 0362-5664 (Letn. 16, št. 6, 1993, str. 550-554)Vrsta gradiva - članek, sestavni delLeto - 1993Jezik - angleškiCOBISS.SI-ID - 10005209
Avtor
Pirtošek, Zvezdan, 1956- |
Merello, Marcelo |
Carlsson, Arvid |
Stern, Gerald
Teme
Parkinson disease |
Drug therapy |
Antiparkinson agents |
Therapeutic use |
Administration and dosage |
Piperidines |
Therapeutic use |
Administration and dosage |
Apomorphine |
Therapeutic use |
Administration and dosage |
Blood pressure |
Drug effects |
Dopamine agonists |
Administration and dosage |
Pharmacology |
Injections, subcutaneous |
Movement |
Drug effects |
Receptors, dopamine d1 |
Agonists |
Receptors, dopamine d2 |
Agonists
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Pirtošek, Zvezdan, 1956- | 05380 |
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