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Stable gastric pentadecapeptide BPC 157-NO-system relationSikirić, Predrag ...We reviewed stable gastric pentadecapeptide BPC 157-NO-system-relation, its close participation in Moncada's (maintained vascular integrity, platelets control) homeostatic healing response of ... NO-system to injury. Namely, BPC 157%s particular healing effect also affects all events after vascular integrity loss (dependent on circumstances, it reduces either thrombosis (abdominal aorta anastomosis) or bleeding/thrombocytopenia (amputation, heparin, warfarin, aspirin)) and in a series of different injurious models, acute and chronic, BPC 157 consistently advances healing after severe injuries in various tissues spontaneously unable to heal; stimulates egr-1 and naB2 genes; exhibits high safety (LD1 not achieved)). Hypothesis, that BPC 157 (since formed constitutively in the gastric mucosa, stable in human gastric juice, along with significance of NO-synthase and the basal formation of NO in stomach mucosa, greater than that seen in other tissues) exhibits a general, effective competing both with L-arginine analogues (i. e., L-NAME) and L-arginine, and that this has some physiologic importance (NO-generation), later, practically supports its beneficial effects illustrating BPC 157 and NOsystem mutual (with L-NAME/L-arginine; alone and together) relations in (i) gastric mucosa and mucosal protection, following alcohol lesions, in cytoprotection course, NO-generation, and blood pressure regulation; (ii) alcohol acute/chronic intoxication, and withdrawal; (iii) cardiovascular disturbances, chronic heart failure, pulmonary hypertension, and arrhythmias; (iv) disturbances after hypokalemia and hyperkalemia, and potassium-cell membrane dysfunction; and finally, in (v) complex healing failure, proved by the fistulas healing, colocutaneous and esophagocutaneous. However, how this advantage of modulating NO-system (i. e., particular effect on eNOS gene), may be practically translated into an enhanced clinical performance remains to be determined.Vir: Current pharmaceutical design. - ISSN 1381-6128 (iss. 7, Vol. 20, 2014, str. 1126-1135)Vrsta gradiva - članek, sestavni del ; neleposlovje za odrasleLeto - 2014Jezik - angleškiCOBISS.SI-ID - 34192857
Avtor
Sikirić, Predrag |
Seiwerth, Sven |
Ručman, Rudolf, 1940- |
Turkovic, Branko |
Stančić-Rokotov, Dinko |
Brčić, Luka |
Sever, Marko, 1981- |
Klicek, Robert |
Radic, Bozo |
Kolenc, Danijela
Teme
arrhythmias |
chronic heart failure |
pentadecapeptide BPC 157 |
aritmije |
kronična srčna odpoved |
pentadekaptid BPC 157
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Baze podatkov, v katerih je revija indeksirana
Ime baze podatkov | Področje | Leto |
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Povezave do osebnih bibliografij avtorjev | Povezave do podatkov o raziskovalcih v sistemu SICRIS |
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Sikirić, Predrag | ![]() |
Seiwerth, Sven | ![]() |
Ručman, Rudolf, 1940- | 09952 |
Turkovic, Branko | ![]() |
Stančić-Rokotov, Dinko | ![]() |
Brčić, Luka | ![]() |
Sever, Marko, 1981- | ![]() |
Klicek, Robert | ![]() |
Radic, Bozo | ![]() |
Kolenc, Danijela | 52857 |
Vir: Osebne bibliografije
in: SICRIS
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