Two Prodrugs of Potent and Selective GluR5 Kainate Receptor Antagonists Actives in Three Animal Models of Pain

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Two Prodrugs of Potent and Selective GluR5 Kainate Receptor Antagonists Actives in Three Animal Models of Pain

Dominguez, Esteban; Iyengar, Smriti; Shannon, Harlan E; Bleakman, David; Alt, Andrew; Arnold, Brian M; Bell, Michael G; Bleisch, Thomas J; Buckmaster, Jennifer L; Castano, Ana M; Del Prado, Miriam; Escribano, Ana; Filla, Sandra A; Ho, Ken H; Hudziak, Kevin J; Jones, Carrie K; Martinez-Perez, Jose A; Mateo, Ana; Mathes, Brian M; Mattiuz, Edward L; Ogden, Ann Marie L; Simmons, Rosa Maria A; Stack, Douglas R; Stratford, Robert E; Winter, Mark A; Wu, Zhipei; Ornstein, Paul L

Journal of medicinal chemistry, 06/2005, Letnik: 48, Številka: 13

Journal Article

Amino acids 5 and 7, two potent and selective competitive GluR5 KA receptor antagonists, exhibited high GluR5 receptor affinity over other glutamate receptors. Their ester prodrugs 6 and 8 were orally active in three models of pain: reversal of formalin-induced paw licking, carrageenan-induced thermal hyperalgesia, and capsaicin-induced mechanical hyperalgesia.

Dostop do baze podatkov JCR je dovoljen samo uporabnikom iz Slovenije. Vaš trenutni IP-naslov ni na seznamu dovoljenih za dostop, zato je potrebna avtentikacija z ustreznim računom AAI.

Leto	Faktor vpliva		Izdaja		Kategorija		Razvrstitev
Leto	JCR	SNIP	JCR	SNIP	JCR	SNIP	JCR	SNIP

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