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Chagasova bolezen in učinkovine za njeno zdravljenje = Chagas disease and drug substances for its treatmentVokič, Nina ; Gomišček, Gregor ; Sollner Dolenc, MarijaChagasova bolezen, ki jo povzroča protozojski parazit Trypanosoma cruzi, predstavlja veliko breme javnega zdravja v Latinski Ameriki in potencialno grožnjo državam po vsem svetu. Okužba, ki se na ... človeka prenese najpogosteje preko okužene stenice, se v najhujši, kronični obliki izrazi kot kardiomiopatija z motnjami srčnega ritma in pojavom srčne odpovedi, nekateri okuženi pa razvijejo prebavne, nevrološke ali mešane spremembe, ki prav tako zahtevajo ustrezno zdravljenje. Kljub dejstvu, da je bila bolezen prvič odkrita že pred več kot sto leti, sta danes za njeno zdravljenje na voljo le dve registrirani zdravili - benznidazol (BNZ) in nifurtimoks (NF), pri čemer velja BNZ za zdravilo prve izbire. Ta učinkovina je nitroimidazolni antiparazitik, ki poleg tega, da pri zdravljenju ne daje zadovoljivih rezultatov, izkazuje tudi številne neželene učinke. Zdravljenje Chagasove bolezni torej več kot očitno predstavlja velik terapevtski izziv, ki so se ga z namenom odkritja učinkovitejših zdravil lotili tako z iskanjem novih tarč, kot tudi z raznimi modifikacijami že registriranih učinkovin. Raziskave so trenutno osredotočene na tri ciljne tarče - CYP51, kruzipain in DNA parazita, kar poleg opisa Chagasove bolezni, njene razširjenosti in trenutnega načina zdravljenja tudi predstavljamo v tem članku.Source: Farmacevtski vestnik : strokovno glasilo slovenske farmacije = pharmaceutical journal of Slovenia. - ISSN 0014-8229 (Letn. 70, št. 3, julij 2019, str. 212-219)Type of material - article, component partPublish date - 2019Language - slovenianCOBISS.SI-ID - 4757105
source: Farmacevtski vestnik : strokovno glasilo slovenske farmacije = pharmaceutical journal of Slovenia. - ISSN 0014-8229 (Letn. 70, št. 3, julij 2019, str. 212-219)
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Database name | Field | Year |
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Links to authors' personal bibliographies | Links to information on researchers in the SICRIS system |
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Vokič, Nina | |
Gomišček, Gregor | 18038 |
Sollner Dolenc, Marija | 08519 |
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