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Balasubramanian, Balu N; St. Laurent, Denis R; Saulnier, Mark G; Long, Byron H; Bachand, Carol; Beaulieu, Francis; Clarke, Wendy; Deshpande, Milind; Eummer, Jeffrey; Fairchild, Craig R; Frennesson, David B; Kramer, Robert; Lee, Frank Y; Mahler, Mikael; Martel, Alain; Naidu, B. Narasimhulu; Rose, William C; Russell, John; Ruediger, Edward; Solomon, Carola; Stoffan, Karen M; Wong, Henry; Zimmermann, Kurt; Vyas, Dolatrai M
Journal of medicinal chemistry, 03/2004, Letnik: 47, Številka: 7Journal Article
A series of fluoroindolocarbazoles were studied with respect to their topoisomerase I activity, cytotoxicity, selectivity, and in vivo antitumor activity. Emerging from this series was BMS-251873, a potential clinical candidate possessing a robust pharmacological profile including curative antitumor activity against prostate carcinoma.
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Leto | Faktor vpliva | Izdaja | Kategorija | Razvrstitev | ||||
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JCR | SNIP | JCR | SNIP | JCR | SNIP | JCR | SNIP |
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Povezave do osebnih bibliografij avtorjev | Povezave do podatkov o raziskovalcih v sistemu SICRIS |
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Vir: Osebne bibliografije
in: SICRIS
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