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  • Discovery of a 2,4-Disubsti...
    Wittman, Mark D; Carboni, Joan M; Yang, Zheng; Lee, Francis Y; Antman, Melissa; Attar, Ricardo; Balimane, Praveen; Chang, Chiehying; Chen, Cliff; Discenza, Lorell; Frennesson, David; Gottardis, Marco M; Greer, Ann; Hurlburt, Warren; Johnson, Walter; Langley, David R; Li, Aixin; Li, Jianqing; Liu, Peiying; Mastalerz, Harold; Mathur, Arvind; Menard, Krista; Patel, Karishma; Sack, John; Sang, Xiaopeng; Saulnier, Mark; Smith, Daniel; Stefanski, Kevin; Trainor, George; Velaparthi, Upender; Zhang, Guifen; Zimmermann, Kurt; Vyas, Dolatrai M

    Journal of medicinal chemistry, 12/2009, Letnik: 52, Številka: 23
    Journal Article

    This report describes the biological activity, characterization, and SAR leading to 9d (BMS-754807) a small molecule IGF-1R kinase inhibitor in clinical development.