Faculty of Pharmacy, Lj. (FFALJ)
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Vpliv odmerka nifedipina za njegovo vezanje na eritrocite = The influence of nifedipine dose on its binding to erythrocytes : diplomska nalogaVolk, UrškaDihidropiridinski blokator kalcijevih kanalèkov nifedipin se uporablja za prepreèevanje in zdravljenje angine pectoris ter za zdravljenje povisanega krvnega tlaka, ker povzroèa dilatacijo arteriol in ... koronarnih zil.Pri svojem delu smo preuèevali vplive hematoloskih parametrov prostovoljcev (hematokrit, koncentracijo hemoglobina, stevilo eritrocitov in levkocitov) na farmakokinetiène parametre (maksimalno plazemsko koncentracijo uèinkovine, èas, v katerem se doseze maksimalna plazemska koncentracija in povrsino pod plazemsko koncentracijsko krivuljo), ki so bili doloèeni po aplikaciji 20 mg pripravka s hitrim sprosèanjem oz. 60 mg pripravka s podaljsanim sprosèanjem. Medsebojne vplive smo statistièno ovrednotili s Pearsonovim koeficientom korelacije in sicer za vse vrednosti farmakokinetiènih parametrov in nato se za vsako podmnozico hematoloskih parametrov posebej. Prav tako smo v 20 oz. 60mg skupini z analizo variance prouèevali vplive hematoloskih parametrov na aritmetiène sredine podmnozic. Z analizo variance smo primerjali tudi srednje vrednosti Pearsonovih koeficientov korelacije znotraj farmakokinetiènih parametrov v 20 oz. 60 mg skupini in tudi posameznih podmnozic znotraj njih. Zmetodo multiple regresije smo za posamezne farmakokinetiène parametre doloèili linearne kombinacije hematoloskih karakteristik, ki so pokazale najmoènejso povezavo oz. najveèji koeficient determinacije. Ugotovili smo, da na farmakokinetiène parametre vpliva vrednost hematokrita, stevilo eritrocitovin koncentracija hemoglobina, neodvisno od odmerka nifedipina. Z eksperimentalnim delom smo potrdili domnevo, da se nifedipin veze na eritrocite, kar se kaze z zmanjsanjem maksimalne plazemske koncentracije in povrsine pod plazemsko koncentracijsko krivuljoType of material - undergr. thesisPublication and manufacture - Ljubljana : [Volk U.], 2001Language - slovenianCOBISS.SI-ID - 953969
Author
Volk, Urška
Other authors
Kozjek, Franc
Topics
nifedipin |
kalcijevi kanalčki |
blokatorji |
farmakologija |
farmakokinetika |
analiza podatkov |
erotrociti |
vezava nifedipina
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Knjižnica dp 0000000615 Volk Urška Vpliv odmerka IN: 0005254 Knjižnica dp 615 Volk Urška Vpliv odmerka IN: 0005254 |
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Knjižnica dp 0000000615 Volk Urška Vpliv odmerka IN: 0005248 Knjižnica dp 615 Volk Urška Vpliv odmerka IN: 0005248 |
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Kozjek, Franc | 00184 |
Source: Personal bibliographies
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